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µå·°ÀÎÆ÷¿¡¼´Â ÀǾàǰ ÀÎÅÍ³Ý ÆÇ¸Å¸¦ ÇÏÁö ¾Ê½À´Ï´Ù. |
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1µî±Þ: ¿øÄ¢Àû »ç¿ë±Ý±â / 2µî±Þ: ¸íÈ®ÇÑ ÀÓ»óÀû ±Ù°Å ¶Ç´Â »çÀ¯°¡ ÀÖ´Â °æ¿ì ºÎµæÀÌÇÏ°Ô »ç¿ë / Mµî±Þ: ÀÓ»óÀû»óȲ¿¡ µû¶ó 1µî±Þ ¶Ç´Â 2µî±ÞÀ¸·Î ºÐ·ùµÇ´Â ¼ººÐ
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20160155 |
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ÀӽŠ2~3±âÁß Åõ¿©½Ã ÅÂ¾Æ ¹× ½Å»ý¾Æ ¼Õ»ó(ÀúÇ÷¾Ð, ½Å±â´ÉºÎÀü, ÇÌ´¢ ±×¸®°í/¶Ç´Â ¹«´¢, ¾ç¼ö°ú¼ÒÁõ, µÎ°³°ñ¹ßÀ°ºÎÀü, Àڱó» ¼ºÀåÁöü), ÆóºÎÀü, ¾È¸éºñÁ¤»ó, »çÁö¿¬Ãà ¹× »ç¸Á °¡´É¼º. |
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1. º»Å°íÇ÷¾Ð
2. ½ÉºÎÀü : Á½ɽǼöÃà±â´ÉÀÌ ¼Õ»óµÈ(NYHA class ¥± ¡ ¥³, Á½ɽǹÚÃâ·ü 40 %ÀÌÇÏ) ½ÉºÎÀü ȯÀÚ Áß ´ÙÀ½¿¡ ÇØ´çÇÏ´Â °æ¿ì
1) ACE¾ïÁ¦Á¦¿¡ ´ëÇÑ Ãß°¡¿ä¹ýÀÌ ÇÊ¿äÇÑ °æ¿ì
2) ACE¾ïÁ¦Á¦¿¡ ³»¾à¼ºÀÌ ÁÁÁö ¾ÊÀº °æ¿ì
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* Àý´ë ÀÓÀǺ¹¿ëÇÏÁö ¸¶½Ã°í ¹Ýµå½Ã ÀÇ»ç ¶Ç´Â ¾à»ç¿Í »ó´ãÇϽñ⠹ٶø´Ï´Ù.
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ÀÌ ¾àÀº ½Ä»ç¿Í °ü°è¾øÀÌ ¸ÅÀÏ ÀÏÁ¤ÇÑ ½Ã°£¿¡ º¹¿ëÇϵµ·Ï ÇÑ´Ù.
1. º»Å°íÇ÷¾Ð
1) ¼ºÀÎ : ÃÊȸ¿ë·® ¹× À¯Áö¿ë·®À¸·Î 1ÀÏ 1ȸ ĵ¥»ç¸£Åº½Ç·º¼¼Æ¿·Î¼ 8 ¡ 16 mg °æ±¸Åõ¿©°¡ ±ÇÀåµÈ´Ù. 1ÀÏ 1ȸ 16 mgÀ¸·Î 4ÁÖ°£ Ä¡·á ÈÄ¿¡µµ Ç÷¾ÐÀÌ ÃæºÐÈ÷ Á¶ÀýµÇÁö ¾Ê´Â °æ¿ì, ÃÖ´ë 1ÀÏ 1ȸ 32 mg±îÁö Áõ·®ÇÒ ¼ö ÀÖ´Ù. ÀÌ ¿ë·®À¸·Îµµ Ç÷¾ÐÀÌ Á¶ÀýµÇÁö ¾Ê´Â °æ¿ì, ´Ù¸¥ Ä¡·á¹ýÀ» °í·ÁÇÏ¿©¾ß ÇÑ´Ù. Ä¡·á°³½Ã 4ÁÖ À̳»¿¡ ÃÖ°íÈ¿°ú°¡ ¹ßÇöµÈ´Ù.
2) °í·ÉÀÚ : Ãʱâ¿ë·®À» Á¶ÀýÇÒ Çʿ䰡 ¾ø´Ù.
3) Ç÷°ü³» À¯È¿Ç÷¾×·® °¨¼Ò(Intravascular volume depletion) ȯÀÚ : À¯È¿ Ç÷¾×·® °¨¼Ò¿Í °°ÀÌ ÀúÇ÷¾ÐÀÇ À§Ç輺ÀÌ ³ôÀº ȯÀÚ¿¡ ´ëÇÏ¿© ¼¼½ÉÇÏ°Ô ÁÖÀÇÇÏ¸é¼ Ãʱâ¿ë·®À¸·Î 4 mgÀ» Åõ¿©ÇÑ´Ù.
4) ½ÅÀå¾Ö ȯÀÚ : Ç÷¾×Åõ¼®È¯ÀÚ¸¦ Æ÷ÇÔÇÑ, ½ÅÀå¾Ö ȯÀÚÀÇ Ãʱâ¿ë·®Àº 4 mgÀ¸·Î, ȯÀÚÀÇ ¹ÝÀÀ¿¡ µû¶ó ¿ë·®À» Á¶ÀýÇÑ´Ù. ÁßÁõ ¶Ç´Â ¸»±â ½ÅÀå¾Ö ȯÀÚ(Å©·¹¾ÆÆ¼´Ñû¼ÒÀ² < 15 mL/min)¿¡ ´ëÇÑ »ç¿ë°æÇèÀÌ Á¦ÇÑÀûÀÌ´Ù.
5) °£Àå¾Ö ȯÀÚ : °æÁõ ¹× Áߵ °£Àå¾Ö ȯÀÚÀÇ Ãʱâ¿ë·®Àº 1ÀÏ 1ȸ 2 mgÀ¸·Î, ȯÀÚÀÇ ¹ÝÀÀ¿¡ µû¶ó ¿ë·®À» Á¶ÀýÇÑ´Ù. ÁßÁõÀÇ °£Àå¾Ö ȯÀÚ¿¡ ´ëÇÑ »ç¿ë°æÇèÀÌ ¾ø´Ù.
6) ¼Ò¾Æ : ¸¸ 18¼¼ ÀÌÇÏÀÇ Ã»¼Ò³â ¹× ¼Ò¾Æ¿¡ ´ëÇÑ ¾ÈÀü¼º ¹× À¯È¿¼ºÀº È®¸³µÇ¾î ÀÖÁö ¾Ê´Ù.
2. ½ÉºÎÀü
1) ¼ºÀÎ : Ãʱâ¿ë·®Àº 1ÀÏ 1ȸ 4 mgÀÌ ±ÇÀåµÈ´Ù. Àû¾îµµ 2ÁÖ ÀÌ»óÀÇ °£°ÝÀ» µÎ°í ¿ë·®À» 2¹è¾¿ Áõ·®Çϸç, ȯÀÚÀÇ ³»¾à¼ºÀ» °í·ÁÇÏ¿© ÃÖ´ë 1ÀÏ 1ȸ 32 mg±îÁö Áõ·®ÇÒ ¼ö ÀÖ´Ù.
2) °í·ÉÀÚ, Ç÷°ü³» À¯È¿Ç÷¾×·® °¨¼ÒȯÀÚ, ½ÅÀå¾Ö ȯÀÚ, °æÁõ ¡ ÁߵÀÇ °£Àå¾ÖȯÀÚ : Ãʱâ¿ë·®À» Á¶ÀýÇÒ Çʿ䰡 ¾ø´Ù.
3) ¼Ò¾Æ : ¸¸ 18¼¼ ÀÌÇÏÀÇ Ã»¼Ò³â ¹× ¼Ò¾Æ¿¡ ´ëÇÑ ¾ÈÀü¼º ¹× À¯È¿¼ºÀº È®¸³µÇ¾î ÀÖÁö ¾Ê´Ù.
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1) ÀÌ ¾à ¶Ç´Â ÀÌ ¾àÀÇ ±¸¼º¼ººÐ¿¡ °ú¹Î¹ÝÀÀ ȯÀÚ
2) ÀӺΠ¶Ç´Â ÀÓ½ÅÇϰí ÀÖÀ» °¡´É¼ºÀÌ ÀÖ´Â ¿©¼º ¹× ¼öÀ¯ºÎ
3) ÁßÁõ °£Àå¾Ö ȯÀÚ ¹×/¶Ç´Â ´ãÁóÁ¤Ã¼ ȯÀÚ
4) À¯Àü¼º Ç÷°üºÎÁ¾ ȯÀÚÀ̰ųª, ACE¾ïÁ¦Á¦ ȤÀº ¾ÈÁö¿ÀÅٽť±¼ö¿ëü ±æÇ×Á¦ Ä¡·á½Ã Ç÷°üºÎÁ¾ÀÇ º´·ÂÀÌ Àִ ȯÀÚ
5) ¿ø¹ß°í¾Ëµµ½ºÅ×·ÐÇ÷Áõ ȯÀÚ(ÀÌ ¾à¹°¿¡ Àß ¹ÝÀÀÇÏÁö ¾Ê´Â´Ù.)
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1) °í·ÉÀÚ
2) °íÄ®·ýÇ÷Áõ ȯÀÚ È¤Àº Ç÷û Ä®·ýÄ¡°¡ ³ô¾ÆÁö±â ½¬¿î ȯÀÚ
3) °æÁõ¿¡¼ Áߵ °£Àå¾Ö ȯÀÚ(¿¹, °£°æº¯ ȯÀÚ)
4) ´ëµ¿¸ÆÆÇ ¹× ½Â¸ðÆÇ ÇùÂøÁõ ȯÀÚ È¤Àº Æó¼âºñ´ë½É±Ùº´ ȯÀÚ
5) ÇãÇ÷ ½ÉÀ庴, ÇãÇ÷ ½ÉÀåÇ÷°ü Áúȯ, ³úÇ÷°ü Àå¾Ö ȯÀÚ(°úµµÇÑ Ç÷¾Ð°ÇÏ´Â ½É±Ù°æ»öÀ̳ª ³úÇ÷·ù ºÎÀüÀ¸·Î ÀÎÇÑ ³úÁ¹ÁßÀ» ÀÏÀ¸Å³ ¼ö ÀÖ´Ù.)
6) ¾çÃø¼º ȤÀº ÆíÃø¼º ½Åµ¿¸Æ ÇùÂøÁõ ȯÀÚ(½ÅÇ÷·ù·®ÀÇ °¨¼Ò³ª »ç±¸Ã¼ ¿©°ú¾ÐÀÇ ÀúÇÏ¿¡ ÀÇÇØ ±Þ¼ÓÈ÷ ½Å±â´ÉÀ» ¾ÇȽÃų ¿ì·Á°¡ ÀÖ´Ù.)
7) Ç÷°ü³» À¯È¿Ç÷¾×·® °¨¼ÒȯÀÚ
8) ½ÅÀå¾Ö ȯÀÚ(°úµµÇÑ °¾Ð¿¡ ÀÇÇØ ½ÅÀå ±â´ÉÀÌ ¾Ç鵃 ¿ì·Á°¡ ÀÖ´Ù.)
9) ÃÖ±Ù ½ÅÀå À̽ÄÀ» ¹ÞÀº ȯÀÚ(»ç¿ë °æÇèÀÌ ¾ø´Ù.)
10) 18¼¼ ¹Ì¸¸ ¼Ò¾Æ ¹× û¼Ò³â
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1) º»Å°íÇ÷¾Ð
ÀϹÝÀûÀ¸·Î ÀÌ»ó¹ÝÀÀÀº °æ¹ÌÇϰí ÀϽÃÀûÀ̾úÀ¸¸ç, ¹ßÇöÀ²Àº ¿ë·®, ¿¬·É, ¼ºº°°ú ¹«°üÇÏ¿´´Ù. ÀÌ»ó¹ÝÀÀÀ¸·Î ÀÎÇØ Ä¡·á¸¦ Áß´ÜÇÏ´Â »ç·Ê´Â ÀÌ ¾à°ú À§¾à±º¿¡¼ À¯»çÇÏ¿´´Ù.
(1) ÀÓ»ó½ÃÇè °á°ú, ĵ¥»ç¸£Åº½Ç·º¼¼Æ¿±º¿¡¼ Àû¾îµµ 1 % ÀÌ»ó ¹ß»ýÇÏ¿´°í À§¾à±º¿¡ ºñÇØ ³ôÀº ºñÀ²·Î ¹ß»ýÇÑ ÀÌ»ó¹ÝÀÀÀº ´ÙÀ½°ú °°´Ù.
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(2) ÀÓ»ó½ÃÇè °á°ú, 1 % ÀÌ»óÀÇ ºñÀ²·Î ¹ß»ýÇÏ¿´Áö¸¸ ÀÌ ¾à¿¡ ºñÇÏ¿© À§¾à Åõ¿©±º¿¡¼ °°°Å³ª ´õ ³ôÀº ºñÀ²·Î ¹ß»ýÇÑ ÀÌ»ó¹ÝÀÀÀº ´ÙÀ½°ú °°´Ù. : ÇÇ·Î, ¸»ÃʺÎÁ¾, ÈäÅë, µÎÅë, ±â°üÁö¿°, ±âħ, ºÎºñ°¿°, ±¸¿ª, º¹Åë, ¼³»ç, ±¸Åä, °üÀýÅë, ´Ü¹é´¢
(3) ÀÓ»ó½ÃÇè °á°ú, ÀÌ ¾à°úÀÇ Àΰú°ü°è¿¡ »ó°ü¾øÀÌ 0.5 % ÀÌ»óÀÇ ¹ß»ýÀ²·Î º¸°íµÈ Áß¿äÇÑ ÀÌ»ó¹ÝÀÀÀº ´ÙÀ½°ú °°´Ù.
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¨ï È£Èí±â°è : È£Èí°ï¶õ
¨ð ÇǺΠ¹× ºÎ¼Ó±â°ü : ¹ßÁø, ¹ßÇÑÁõ°¡
¨ñ ºñ´¢±â°è : Ç÷´¢
2) ½ÉºÎÀü
½ÉºÎÀü ȯÀÚ¿¡¼ÀÇ ÀÌ»ó¹ÝÀÀ ¹ßÇö¾ç»óÀº ¾à¸®ÀÛ¿ë ¹× È¯ÀÚÀÇ °Ç°»óÅÂ¿Í ÀÏÄ¡ÇÏ¿´´Ù. ÀÌ ¾à 32 mg(n=3,803)±º°ú À§¾à(n=3,796)±ºÀ» ºñ±³ÇÑ CHARM ÀÓ»ó½ÃÇè¿¡¼ ÀÌ ¾à Åõ¿©±ºÀÇ 21.0 %, À§¾à±ºÀÇ 16.1 %°¡ ÀÌ»ó¹ÝÀÀÀ¸·Î ÀÎÇÏ¿© Åõ¿©¸¦ Áß´ÜÇÏ¿´´Ù. ÀÚÁÖ(¡Ã 1/100, < 1/10) ³ªÅ¸³ ÀÌ»ó¹ÝÀÀÀº ÀúÇ÷¾Ð, °íÄ®·ýÇ÷Áõ, ½Å±â´É ¼Õ»ó, Å©·¹¾ÆÆ¼´Ñ, ¿ä¼Ò, Ä®·ýÀÇ Áõ°¡¿´´Ù. ¿ë·®À» Áõ°¡ÇÏ´Â µ¿¾È°ú ±× ÀÌÈÄ Á¤±âÀûÀ¸·Î Ç÷ûĮ·ý°ú Å©·¹¾ÆÆ¼´Ñ ¼öÄ¡¸¦ ¸ð´ÏÅ͸µ ÇÏ´Â °ÍÀÌ ±ÇÀåµÈ´Ù.
3) ÀϹÝÀûÀ¸·Î ÀÌ ¾àÀº ÀÏ»óÀûÀÎ ½ÇÇè½ÇÀû ÀÎÀڵ鿡 ÀÓ»óÀûÀ¸·Î À¯ÀÇÇÒ¸¸ÇÑ ¿µÇâÀ» ¹ÌÄ¡Áö ¾Ê¾Ò´Ù. ´Ù¸¥ ·¹´Ñ-¾ÈÁö¿ÀÅÙ½Å-¾Ëµµ½ºÅ×·Ð°è ¾ïÁ¦Á¦¿Í ¸¶Âù°¡Áö·Î Çì¸ð±Û·Îºó°ú Ç츶ÅäÅ©¸®Æ®Ä¡°¡ ¾à°£ °¨¼ÒÇÏ¿´´Ù. Å©·¹¾ÆÆ¼´Ñ, ¿ä¼Ò, Ä®·ýÀÇ Áõ°¡¿Í ³ªÆ®·ýÀÇ °¨¼Ò°¡ °üÂûµÇ¾ú´Ù. ÀÌ»ó¹ÝÀÀÀ¸·Î ALTÀÇ »ó½ÂÀÌ ÀÌ ¾à Åõ¿©±º¿¡¼ À§¾à±º¿¡ ºñÇØ ¾à°£ ³ôÀº ºóµµ·Î º¸°íµÇ¾ú´Ù(1.3 % vs 0.5 %). ÀÌ ¾àÀ» Åõ¿© ¹ÞÀº ȯÀÚ¿¡¼ ½ÇÇè½ÇÀû ÀÎÀÚµéÀÇ ÀÏ»óÀûÀÎ ¸ð´ÏÅ͸µÀº ÇÊ¿äÇÏÁö ¾ÊÀ¸³ª, ½Å±â´É ¼Õ»óÀÚ¿¡¼´Â Ç÷ûĮ·ý°ú Å©·¹¾ÆÆ¼´Ñ ¼öÄ¡¸¦ Á¤±âÀûÀ¸·Î ¸ð´ÏÅ͸µ ÇÏ´Â °ÍÀÌ ±ÇÀåµÈ´Ù.
4) ½ÃÆÇ ÈÄ Á¶»ç¿¡¼ ¸Å¿ì µå¹°°Å³ª(< 1/10,000) ºóµµ¸¦ ¾Ë ¼ö ¾ø°Ô ³ªÅ¸³ ÀÌ»ó¹ÝÀÀÀº ´ÙÀ½°ú °°´Ù.
(1) Ç÷¾× ¹× ¸²ÇÁ°è : ¹éÇ÷±¸°¨¼ÒÁõ, È£Áß±¸°¨¼ÒÁõÀÌ ³ªÅ¸³¯ ¼ö ÀÖ´Ù. ¶ÇÇÑ ¹«°ú¸³±¸ÁõÀÌ ³ªÅ¸³¯ ¼ö ÀÖÀ¸¹Ç·Î °üÂûÀ» ÃæºÐÈ÷Çϰí ÀÌ»óÀÌ ÀÎÁ¤µÇ´Â °æ¿ì¿¡´Â Åõ¿©¸¦ ÁßÁöÇϰí ÀûÀýÇÑ Ã³Ä¡¸¦ ÇÑ´Ù.
(2) ´ë»ç ¹× ¿µ¾çÀÌ»ó : °íÄ®·ýÇ÷Áõ, Àú³ªÆ®·ýÇ÷Áõ, ÀúÇ÷´ç(´ç´¢º´ Ä¡·á ÁßÀΠȯÀÚ¿¡¼ ³ªÅ¸³ª±â ½±´Ù.)ÀÌ ³ªÅ¸³¯ ¼ö ÀÖÀ¸¹Ç·Î °üÂûÀ» ÃæºÐÈ÷ Çϰí, ¹«·Â°¨, °øº¹°¨, ½ÄÀº¶¡, ¼Õ ¶³¸², ÁýÁß·Â ÀúÇÏ, °æ·Ã, ÀÇ½Ä Àå¾Ö µîÀÌ ³ªÅ¸³ °æ¿ì ¿¡´Â Åõ¿©¸¦ ÁßÁöÇϰí ÀûÀýÇÑ Ã³Ä¡¸¦ ÇÑ´Ù.
(3) ½Å°æ°è : ¾îÁö·³, µÎÅëÀÌ ³ªÅ¸³¯ ¼ö ÀÖ´Ù.
(4) ¼Òȱâ°è : ±¸¿ª, ¼³»ç°¡ ³ªÅ¸³¯ ¼ö ÀÖ´Ù.
(5) °£´ãµµ°è : °£ È¿¼ÒÄ¡ Áõ°¡, °£¿°ÀÌ ³ªÅ¸³¯ ¼ö ÀÖ´Ù. ¶ÇÇÑ AST, ALT, ¥ã-GTP »ó½Â µîÀÇ °£±â´É Àå¾Ö, Ȳ´ÞÀÌ ³ªÅ¸³¯ ¼ö ÀÖÀ¸¹Ç·Î °üÂûÀ» ÃæºÐÈ÷Çϰí ÀÌ»óÀÌ ÀÎÁ¤µÇ´Â °æ¿ì¿¡´Â Åõ¿©¸¦ ÁßÁöÇϰí ÀûÀýÇÑ Ã³Ä¡¸¦ÇÑ´Ù.
(6) ÇǺΠ¹× ÇÇÇÏÁ¶Á÷ : ¹ßÁø, µÎµå·¯±â, °¡·Á¿òÁõÀÌ ³ªÅ¸³¯ ¼ö ÀÖ´Ù. ¶ÇÇÑ Ç÷°üºÎÁ¾(¾ó±¼, ±¸¼ø¡¤Çô, ÀΡ¤ÈĵΠµîÀÇ Á¾Ã¢)ÀÌ ³ªÅ¸³¯ ¼ö ÀÖÀ¸¹Ç·Î °üÂûÀ» ÃæºÐÈ÷ Çϰí ÀÌ»óÀÌ ÀÎÁ¤µÇ´Â °æ¿ì¿¡´Â Åõ¿©¸¦ ÁßÁöÇϰí ÀûÀýÇÑ Ã³Ä¡¸¦ ÇÑ´Ù.
(7) ±ÙÀ°Åë, ¹«·Â°¨, Å©·¹¾ÆÆ¾Å°³ª¾ÆÁ¦(CK) »ó½Â, Ç÷Áß ¹× ¿äÁß ¹Ì¿À±Û·Îºó »ó½ÂÀ» Ư¡À¸·Î Çϴ Ⱦ¹®±ÙÀ¶Çذ¡ ³ªÅ¸³¯ ¼ö ÀÖÀ¸¹Ç·Î °üÂûÀ» ÃæºÐÈ÷Çϰí ÀÌ·¯ÇÑ °æ¿ì¿¡´Â Åõ¿©¸¦ ÁßÁöÇϰí ÀûÀýÇÑ Ã³Ä¡¸¦ ÇÑ´Ù.
(8) ±Ù°ñ°Ý°è : °üÀýÅë, ±ÙÀ°Åë, ¿äÅëÀÌ ³ªÅ¸³¯ ¼ö ÀÖ´Ù.
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(1) ÁßÃß ¹× ¸»ÃʽŰæ°è : ¸¶ºñ(2¸í), ±äÀåÇ×Áø(1¸í)
(2) Àü½Å : ½Ç½Å(1¸í), ¾ó±¼È«Á¶(1¸í), üÁßÁõ°¡(1¸í), ¾ó±¼ºÎÁ¾(1¸í)
(3) À§Àå°ü°è : ±¸°¥(2¸í)
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(5) °¨°¢±â°ü : À̸í(1¸í), ¹Ì°¢µµÂø(1¸í)
(6) »ý½Ä±â°è : ¹ß±âºÎÀü(1¸í)
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1) ÀÓ»óÀû À¯ÀǼº ÀÖ´Â ¾à¹°»óÈ£ÀÛ¿ëÀº º¸°íµÈ ¹Ù ¾ø´Ù. ÀÓ»ó ¾àµ¿ÇÐ ¿¬±¸¿¡¼ Á¶»çµÈ ¹°ÁúµéÀº È÷µå·ÎŬ·Î·ÎƼ¾ÆÁöµå, ¿Í¸£ÆÄ¸°, µð°î½Å, °æ±¸¿ëÇÇÀÓ¾à(Áï, ¿¡Æ¼´Ò¿¡½ºÆ®¶óµð¿Ã/·¹º¸³ë¸£°Ô½ºÆ®·¼), ±Û¸®º¥Å¬¶ó¹Ìµå, ´ÏÆäµðÇÉ µîÀÌ´Ù.
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3) ÀÌ ¾àÀÇ Ç÷¾Ð°ÇÏÈ¿°ú´Â ´Ù¸¥ Ç÷¾Ð°ÇÏÁ¦¿¡ ÀÇÇØ »ó½ÂµÉ ¼öµµ ÀÖ´Ù.
4) ACE¾ïÁ¦Á¦¿Í ¸®Æ¬À» º´¿ëÇßÀ» ¶§, Ç÷û ¸®Æ¬³óµµ ¹× µ¶¼ºÀÌ °¡¿ªÀûÀ¸·Î Áõ°¡µÇ¾ú´Ù. À¯»çÇÑ È¿°ú°¡ ¾ÈÁö¿ÀÅٽť±¼ö¿ëü ±æÇ×Á¦¿¡¼ ³ªÅ¸³¯ ¼ö ÀÖÀ¸¹Ç·Î Ç÷û ¸®Æ¬¼öÄ¡¸¦ ÁÖÀDZí°Ô ¸ð´ÏÅ͸µ ÇÏ´Â °ÍÀÌ ±ÇÀåµÈ´Ù.
5) ¾ÈÁö¿ÀÅٽť±¼ö¿ëü ±æÇ×Á¦°¡ ºñ½ºÅ×·ÎÀ̵å¼Ò¿°ÁøÅëÁ¦(¿¹, ¼±ÅÃÀûÀÎ COX-2¾ïÁ¦Á¦, ¾Æ¼¼Æ¿»ì¸®½Ç»ê(> 3 g/day), ºñ¼±ÅÃÀû ºñ½ºÅ×·ÎÀ̵å¼Ò¿°ÁøÅëÁ¦)¿Í º´¿ë ½Ã Ç÷¾Ð°ÇÏÈ¿°ú°¡ °¨¼ÒÇÒ ¼ö ÀÖ´Ù. ACE¾ïÁ¦Á¦¿Í °°ÀÌ, ¾ÈÁö¿ÀÅٽť±¼ö¿ëü ±æÇ×Á¦¿Í ºñ½ºÅ×·ÎÀ̵å¼Ò¿°ÁøÅëÁ¦ÀÇ º´¿ëÀº ½Å±â´ÉÀ» ¾ÇÈ, ±Þ¼º ½ÅºÎÀüÀ» À¯¹ß½Ãų ¼ö ÀÖ°í, Ç÷û Ä®·ýÀ» Áõ°¡½Ãų ¼ö ÀÖ´Ù. º´¿ë½Ã ÁÖÀÇÇØ¾ß Çϸç, ƯÈ÷ °í·ÉÀÚ È¤Àº À¯È¿Ç÷¾×·® °¨¼ÒȯÀÚ(ÀÌ´¢Á¦ Ä¡·á ÁßÀΠȯÀÚ¸¦ Æ÷ÇÔ)´Â ÁÖÀÇÇÑ´Ù. º´¿ëÄ¡·á ½ÃÀÛ ÈÄ¿¡ ȯÀÚ¿¡°Ô ÀûÀýÇÑ ¼öºÐÀÌ °ø±ÞµÇ¾î¾ß Çϸç, ½Å±â´ÉÀ» ÁÖ±âÀûÀ¸·Î ¸ð´ÏÅ͸µ ÇØ¾ßÇÑ´Ù.
6) ·¹´Ñ-¾ÈÁö¿ÀÅÙ½Å-¾Ëµµ½ºÅ׷а迡 ¿µÇâÀ» ¹ÌÄ¡´Â ´Ù¸¥ Á¦Á¦ÀÇ »ç¿ë°æÇè¿¡ ±Ù°ÅÇØ º¼ ¶§ ÀÌ ¾à°ú Ä®·ýº¸ÀüÀÌ´¢Á¦(½ºÇǷγë¶ôÅæ, Æ®¸®¾ÏÅ×·» µî), Ä®·ýº¸ÃæÁ¦, Ä®·ýÀ» ÇÔÀ¯ÇÏ´Â ¿°º¸ÃæÁ¦ ¶Ç´Â Ä®·ý¼öÄ¡¸¦ Áõ°¡½Ãų ¼ö ÀÖ´Â ´Ù¸¥ Á¦Á¦µé(¿¹, ÇìÆÄ¸°)°ú º´¿ëÅõ¿©ÇÒ °æ¿ì Ç÷ûĮ·ý³óµµ°¡ Áõ°¡ÇÒ ¼ö ÀÖÀ¸¹Ç·Î ÁÖÀÇÇϵµ·Ï ÇÑ´Ù.
7) ÀÌ ¾àÀÇ »ýüÀÌ¿ë·üÀº À½½Ä¹°¿¡ ÀÇÇØ ¿µÇâÀ» ¹ÞÁö ¾Ê´Â´Ù.
8) ACE¾ïÁ¦Á¦ È¿°ú°¡ ºÒÃæºÐÇÑ È¯ÀÚ¿¡°Ô ÀÌ ¾àÀÇ À¯È¿¼º ¹× ¾ÈÀü¼º, ±×¸®°í ACE¾ïÁ¦Á¦¿Í º´¿ëÅõ¿©½Ã ÀÌ ¾àÀÇ À¯È¿¼º ¹× ¾ÈÀü¼ºÀº È®¸³µÇÁö ¾Ê¾Ò´Ù. ½ÉºÎÀü ȯÀÚ¿¡¼ ACE¾ïÁ¦Á¦¿Í º´¿ë½Ã ½Å±â´ÉÀå¾Ö¿Í °íÄ®·ýÇ÷Áõ°ú °°Àº ÀÌ»ó¹ÝÀÀÀÇ À§ÇèÀÌ Áõ°¡ÇÑ´Ù. µû¶ó¼ º´¿ë ½Ã ÁÖÀÇÇØ¾ß ÇÑ´Ù.
9) ÀÌ ¾à°ú ¾Æ¼¼³ëÄڿ츶·Ñ ȤÀº ÆæÇÁ·ÎÄÚ¿ì¸ó°úÀÇ »óÈ£ÀÛ¿ëÀº ¿¬±¸µÈ ¹Ù°¡ ¾øÀ¸¹Ç·Î, À§¿Í °°Àº Ç×ÀÀ°íÁ¦¿Í ÀÌ ¾àÀº º´¿ë ½Ã ÁÖÀÇÇØ¾ß ÇÑ´Ù.
10) ACE¾ïÁ¦Á¦, Ä®·ýº¸ÀüÀÌ´¢Á¦, ±×¸®°í ÀÌ ¾àÀÇ º´¿ëÀº ±ÇÀåµÇÁö ¾Ê´Â´Ù.
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(D in 2'nd and 3'rd trimesters )
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»ó±â ÀÓºÎÅõ¿©¿¡ ´ëÇÑ Á¤º¸´Â Àü»êó¸® µÇ¸é¼ ÀÔ·Â ¿À·ù °¡´É¼ºÀÌ Á¸ÀçÇÕ´Ï´Ù. ¿À·ù °¡´É¼ºÀ» ÃÖ¼ÒÈÇϱâ À§ÇÏ¿© ¸¹Àº ³ë·ÂÀ» ±â¿ïÀ̰í ÀÖÀ¸³ª, ±× Á¤È®¼º¿¡ ´ëÇÏ¿© È®½ÅÀ» µå¸± ¼ö ¾ø½À´Ï´Ù. ÀÌ¿¡ ´ëÇØ ȸ»ç´Â Ã¥ÀÓÀ» ÁöÁö ¾Ê½À´Ï´Ù.
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| Ç׸ñ |
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| DUR (ÀǾàǰ»ç¿ëÆò°¡) |
º´¿ë±Ý±â :
°í½ÃµÈ º´¿ë±Ý±â ³»¿ëÀº ¾ø½À´Ï´Ù.
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| Mechanism of Action |
Candesartan¿¡ ´ëÇÑ Mechanism_Of_Action Á¤º¸ Candesartan competes with angiotensin II for binding at the AT1 receptor subtype. As angiotensin II is a vasoconstrictor which also stimulates the synthesis and release of aldosterone, blockage of its effects results in a decreases in systemic vascular resistance.
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| Pharmacology |
Candesartan¿¡ ´ëÇÑ Pharmacology Á¤º¸ Candesartan, a specific angiotensin II antagonist, is used alone or with other antihypertensive agents to treat hypertension. Unlike the angiotensin receptor antagonist losartan, Candesartan does not have an active metabolite or possess uricosuric effects.
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| Metabolism |
Candesartan¿¡ ´ëÇÑ Metabolism Á¤º¸ # Phase_1_Metabolizing_Enzyme:Cytochrome P450 11B2 (CYP11B2)
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| Protein Binding |
Candesartan¿¡ ´ëÇÑ ´Ü¹é°áÇÕ Á¤º¸ Candesartan is highly bound to plasma proteins (>99%) and does not penetrate red blood cells.
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| Half-life |
Candesartan¿¡ ´ëÇÑ ¹Ý°¨±â Á¤º¸ Approximately 9 hours.
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| Absorption |
Candesartan¿¡ ´ëÇÑ Absorption Á¤º¸ Following administration of the candesartan cilexetil prodrug, the absolute bioavailability of candesartan was estimated to be 15%. Food with a high fat content has no affect on the bioavailability of candesartan from candesartan cilexetil.
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| Pharmacokinetics |
Candesartan cilexetilÀÇ ¾à¹°µ¿·ÂÇÐÀÚ·á
- ¾àÈ¿ ¹ßÇö½Ã°£ : 2-4½Ã°£
- ÃÖ°í È¿°ú ¹ßÇö½Ã°£ : 6-8 ½Ã°£
- ÃÖ°í Ç÷Áß³óµµ µµ´Þ½Ã°£ : 3-4 ½Ã°£
- ¾àÈ¿ Áö¼Ó½Ã°£ : 24½Ã°£ ÀÌ»ó
- »ýü³»ÀÌ¿ë·ü : 15%, À½½Ä¹°¿¡ ÀÇÇØ ¿µÇâÀ» ¹ÞÁö ¾ÊÀ½
- ºÐÆ÷¿ëÀû : 0.13 L/kg
- ´Ü¹é°áÇÕ : 99 % ÀÌ»ó
- ´ë»ç : Candesartan cilexetilÀº Èí¼ö°úÁ¤¿¡¼ 99% ÀÌ»óÀÌ À§Àå°ü º®¿¡¼ Ȱ¼ºÇü ´ë»çüÀÎ candesartanÀ¸·Î ´ë»çµÊ
- ¹Ý°¨±â : CandesartanÀ¸·Î 5.1-10.5 ½Ã°£
- ¼Ò½Ç : CandesartanÀº °ÅÀÇ ¹Ìº¯Èü·Î 67% ´ëº¯, 33% ´¢¹è¼³
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| Biotransformation |
Candesartan¿¡ ´ëÇÑ Biotransformation Á¤º¸ During absorption from the gastrointestinal tract, the prodrug candesartan cilexetil undergoes rapid and complete ester hydrolysis to form the active drug, candesartan. Elimination of candesartan is primarily as unchanged drug in the urine and, by the biliary route, in the feces. Minor hepatic metabolism of candesartan occurs by O -deethylation to form an inactive metabolite.
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| Toxicity |
Candesartan¿¡ ´ëÇÑ Toxicity Á¤º¸ No lethality was observed in acute toxicity studies in mice, rats and dogs given single oral doses of up to 2000 mg/kg of candesartan cilexetil or in rats given single oral doses of up to 2000 mg/kg of candesartan cilexetil in combination with 1000 mg/kg of hydrochlorothiazide. In mice given single oral doses of the primary metabolite, candesartan, the minimum lethal dose was greater than 1000 mg/kg but less than 2000 mg/kg.
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| Drug Interactions |
Candesartan¿¡ ´ëÇÑ Drug_Interactions Á¤º¸ Amiloride Increased risk of hyperkaliemiaDrospirenone Increased risk of hyperkaliemiaLithium The ARB increases serum levels of lithiumPotassium Increased risk of hyperkaliemiaSpironolactone Increased risk of hyperkaliemiaTriamterene Increased risk of hyperkaliemia
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CYP450 Drug Interaction |
[CYP450 TableÁ÷Á¢Á¶È¸]
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| Food Interaction |
Candesartan¿¡ ´ëÇÑ Food Interaction Á¤º¸ Take without regard to meals.Administer on a regular basis, at about the same time each day.
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| Drug Target |
[Drug Target]
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| Description |
Candesartan¿¡ ´ëÇÑ Description Á¤º¸ Candesartan, a specific angiotensin II antagonist, is used alone or with other antihypertensive agents to treat hypertension. Candesartan competes with angiotensin II for binding at the AT1 receptor subtype. As angiotensin II is a vasoconstrictor which also stimulates the synthesis and release of aldosterone, blockage of its effects results in a decreases in systemic vascular resistance.
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| Dosage Form |
Candesartan¿¡ ´ëÇÑ Dosage_Form Á¤º¸ Tablet Oral
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| Drug Category |
Candesartan¿¡ ´ëÇÑ Drug_Category Á¤º¸ Angiotensin II Receptor AntagonistsAngiotensin II Type 1 Receptor BlockersAntihypertensive Agents
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| Smiles String Canonical |
Candesartan¿¡ ´ëÇÑ Smiles_String_canonical Á¤º¸ CCOC1=NC2=CC=CC(C(O)=O)=C2N1CC1=CC=C(C=C1)C1=CC=CC=C1C1=NNN=N1
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| Smiles String Isomeric |
Candesartan¿¡ ´ëÇÑ Smiles_String_isomeric Á¤º¸ CCOC1=NC2=CC=CC(C(O)=O)=C2N1CC1=CC=C(C=C1)C1=CC=CC=C1C1=NNN=N1
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| InChI Identifier |
Candesartan¿¡ ´ëÇÑ InChI_Identifier Á¤º¸ InChI=1/C24H20N6O3/c1-2-33-24-25-20-9-5-8-19(23(31)32)21(20)30(24)14-15-10-12-16(13-11-15)17-6-3-4-7-18(17)22-26-28-29-27-22/h3-13H,2,14H2,1H3,(H,31,32)(H,26,27,28,29)/f/h28,31H
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| Chemical IUPAC Name |
Candesartan¿¡ ´ëÇÑ Chemical_IUPAC_Name Á¤º¸ 2-ethoxy-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]benzimidazole-4-carboxylic acid
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