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3) Á¤½Å½Å°æ°è : ¸ðµç Åõ¿©¿ë·®¿¡¼ ºÒÄè°¨ÀÌ ³ªÅ¸³¯ ¼ö ÀÖ°í, Áßµ¶¼ºÁ¤½Åº´µµ º¸°íµÇ¾ú´Ù. Á¹¸², ÀÌ»óȲȦ°¨, ºÒ¾È, ÀÌÁúÅë, Åë°¢°ú¹Î, ´ÙÇÑÁõÀÌ ³ªÅ¸³¯ ¼ö ÀÖ°í, µå¹°°Ô ¼ö¸·°³» Ä«Å×ÅÍ »ðÀÔÀ¸·Î ÀÎÇÑ µÎÅëÀÌ ¸çÄ¥°£ ³ªÅ¸³¯ ¼ö Àִµ¥, Åë»óÀûÀÎ ¹æ¹ýÀ¸·Î óġÇÑ´Ù.
4) °ú¹Î¹ÝÀÀ : °æ¸·¿Ü ¶Ç´Â ¼ö¸·°³» ´Üȸ Åõ¿© ½Ã ³ôÀº ºóµµ·Î °¡·Á¿òÀÌ ³ªÅ¸³ª´Âµ¥, ÀÌ´Â Åõ¿© ¿ë·®°ú °ü·ÃÀÌ ÀÖÀ¸³ª, Åõ¿© ºÎÀ§¿¡¸¸ ±¹ÇѵÇÁö´Â ¾Ê´Â´Ù. ¹®Çå»ó °æ¸·¿Ü ¶Ç´Â ¼ö¸·°³» ¿¬¼ÓÅõ¿© ½Ã °¡·Á¿òÀÌ º¸°íµÇ¾ú´Âµ¥, ±× ¿øÀÎÀº ¾Ë·ÁÁ® ÀÖÁö ¾Ê´Ù. µÎµå·¯±â, ¹ßÁø, ±¹¼ÒÁ¶Á÷ÀڱعÝÀÀÀÌ ³ªÅ¸³¯ ¼ö ÀÖ´Ù.
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6) ¼Òȱâ°è : ±¸¿ª, ±¸Åä°¡ ³ªÅ¸³¯ ¼ö Àִµ¥, Àú¿ë·®(0.2 mg)ÀÇ ³¯·Ï¼Õ Åõ¿©·Î Áõ»óÀ» °æ°¨½Ãų ¼ö ÀÖ´Ù. º¯ºñ, ´ãµµ°æ·Ã, ±¸°°ÇÁ¶, ÃéÀå¿°, ¿Àµð °ý¾à±Ù ¿¬Ãà µîÀÌ ³ªÅ¸³¯ ¼ö ÀÖ´Ù.
7) ±âŸ : ¿¬¼ÓÁÖÀÔÀåÄ¡ »ðÀÔ¼ú ÈÄ ¿øÀκҸíÀÇ ¸»ÃʺÎÁ¾(³²¼º »ý½Ä±â ºÎÁ¾ Æ÷ÇÔ)ÀÌ º¸°íµÇ¾ú´Ù. ±Þ¼º Àü½Å¹ßÁø³óÆ÷Áõ(AGEP), ÁßÃß¼º ¼ö¸é ¹«È£Èí ÁõÈıº, ±âħ¹Ý»ç ¾ïÁ¦, ü¿ÂÁ¶Àý Àå¾Ö°¡ ³ªÅ¸³¯ ¼ö ÀÖ´Ù.
8) ±¹³» ÀÚ¹ßÀû À¯ÇØ»ç·Ê º¸°íÀÚ·á(1989-2013 »ó¹Ý±â)¸¦ ºÐ¼®ÇÑ °á°ú, À¯ÇØ»ç·Ê°¡ º¸°íµÈ ´Ù¸¥ ÀǾàǰ¿¡¼ ¹ß»ýÇÑ À¯ÇØ»ç·Ê¿¡ ºñÇØ Åë°èÀûÀ¸·Î À¯ÀÇÇÏ°Ô ¸¹ÀÌ º¸°íµÈ À¯ÇØ»ç·Ê´Â ´ÙÀ½°ú °°ÀÌ ³ªÅ¸³µ´Ù. ´Ù¸¸, À̷μ °ð ÇØ´ç¼ººÐ°ú ´ÙÀ½ÀÇ À¯ÇØ»ç·Ê °£¿¡ Àΰú°ü°è°¡ ÀÔÁõµÈ °ÍÀ» ÀǹÌÇÏ´Â °ÍÀº ¾Æ´Ï´Ù.
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3) ÀÌ ¾à°ú °°Àº ¾ÆÆí¾ç ¼ö¿ëüÀÇ ¿ÏÀüÈ¿ÇöÁ¦¸¦ Åõ¿©¹Þ°í Àִ ȯÀÚ¿¡°Ô ÆæÅ¸Á¶½Å, ³¯ºÎÇÉ, ºÎÇÁ·¹³ë¸£ÇÉ µîÀÇ ¾ÆÆí¾ç ¼ö¿ëüÀÇ ºÎºÐÈ¿ÇöÁ¦¸¦ Åõ¿©Çϸé, °æÀïÀû ¼ö¿ëü Â÷´ÜÀ¸·Î ÀÎÇØ ÀÌ ¾àÀÇ ÁøÅë È¿°ú¸¦ °¨¼Ò½ÃŰ°Å³ª ±Ý´ÜÁõ»óÀ» ÃËÁø½Ãų ¼ö ÀÖÀ¸¹Ç·Î º´¿ëÅõ¿©ÇÏÁö ¾Ê´Â´Ù.
4) ÀÌ ¾à°ú ½Ã¸ÞƼµòÀÇ Àå±â º´¿ëÅõ¿© ½Ã ÀÌ ¾àÀÇ Ç÷Áß³óµµ°¡ Áõ°¡µÉ ¼ö ÀÖ´Ù.
5) Ç÷Áß ¸ð¸£ÇÉ ³óµµ´Â ¸®ÆÊÇǽſ¡ ÀÇÇØ °¨¼ÒÇÒ ¼ö ÀÖ´Ù. ¸®ÆÊÇǽÅÀ¸·Î Ä¡·áÇÏ´Â µ¿¾È ±×¸®°í Ä¡·áÇÑ ÀÌÈÄ¿¡ ¸ð¸£ÇÉÀÇ ÁøÅë È¿°ú¸¦ ¸ð´ÏÅ͸µÇÏ°í ¿ë·®À» Á¶ÀýÇØ¾ß ÇÑ´Ù.
6) °æ±¸¿ë P2Y12¾ïÁ¦Á¦(¿¹, Ŭ·ÎÇǵµ±×·¼, ÇÁ¶ó¼ö±×·¼, Ƽī±×·¼·¯)¿Í ¸ð¸£ÇɰúÀÇ º´¿ëÅõ¿©´Â °æ±¸¿ë P2Y12¾ïÁ¦Á¦ÀÇ Èí¼ö¿Í ÃÖ°í³óµµ °¨¼Ò ¹× Ç×Ç÷¼ÒÆÇ È¿°ú¸¦ Áö¿¬ÇÒ ¼ö ÀÖ´Ù.
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8. Æó»ö¼º Ç÷ÀüÇ÷°ü¿°(Buerger's disease)À¸·Î 1ÀÏ ¼öȸ ³»¿øÇÏ¿©Àå±â Åõ¿©ÇÑ ¸ôÇÉ(ÁÖ) ¹× ÁøÂû·á ÀÎÁ¤¿©ºÎ
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P.I) 1³âÀü Burger's disease Áø´Ü, »ó±â C.C·Î ÁøÅëÁ¦ ¸Â±â ¿øÇØ ER ³»¿ø.
Tx.) Demerol 1¨Í IM.
ÀÌÈÄ ¿Ü·¡ Áø·á±â·Ï¿¡ Áø·áÀÏ ±â·ÏÀÌ ¾ø¾î ÃÖÃÊ Morphine Åõ¿©ÀÏ È®ÀξȵÊ. Ÿ¾àÁ¦ »ç¿ë³»¿ª ¾øÀ¸¸ç ÇÏ·ç 1-2ȸ ¿Ü·¡ ¹æ¹®ÇÏ¿© Morphine 1.5¨ÍÀ» IV ¶Ç´Â IM(ÁÖ·Î IV)À¸·Î°è¼Ó Åõ¿© ¹Þ¾ÒÀ½.
'02.2.14 2nd fingerpus collection ¼Ò°ß°úÇÔ²² distal phalanx shrinkage ¼Ò°ßº¸¿© woundrevision ¸îÂ÷·ÊÇßÀ¸³ª ¿ÀÈÄ, ¹ã¿¡ ¹«´Ü¿ÜÃâ °è¼ÓÇϰí ÀÖÀ¸¸ç Morphine addictionÀ¸·Î injection Åõ¿© °è¼Ó ¿øÇÔ. injection refuseÇÏ¸é ±ØµµÀÇ ÈïºÐ»óÅ º¸¿© º´½Ç°ú ¿Ü·¡¿¡¼ ÇàÆÐºÎ¸®´Â ¸ð½À º¸ÀÓ. º¸È£ÀÚ¿¡°Ô Áßµ¶¾ç»ó ¼³¸íÇÏ°í °Ý¸®Ä¡·á ¼³¸íÇßÀ¸³ª ȯÀÚ °ÅÀýÇϰí ÀÖÀ½.
'03.11.2 Morphine 15§·¡¿3, NSAID¹× ´Ù¸¥ ÁøÅëÁ¦·Î pain controlÇØº¸ÀÚ°í 30ºÐÀ̻󼳸í»ó´ãÇßÀ¸³ª °áÄÚ ´Ù¸¥ ÁÖ»ç´Â ¾Èµè´Â´ÙÇÏ¿© Morphine Åõ¿©ÇÔ.
29 Chestpain, vomitingÀ¸·Î ÀÀ±Þ½Ç ³»¿ø ¡æ NTG È¿°ú¾øÀ½, Morphine10§·Åõ¿©ÈÄ Áõ»ó »ç¶óÁü. ÀÌÈÄ 15§·¾¿ 3ȸ ´õ Åõ¿©ÇÔ.
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Morphine¿¡ ´ëÇÑ Mechanism_Of_Action Á¤º¸ The precise mechanism of the analgesic action of morphine is unknown. However, specific CNS opiate receptors have been identified and likely play a role in the expression of analgesic effects. The mechanism of respiratory depression involves a reduction in the responsiveness of the brain stem respiratory centers to increases in carbon dioxide tension and to electrical stimulation.
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| Pharmacology |
Morphine¿¡ ´ëÇÑ Pharmacology Á¤º¸ Morphine is a narcotic pain management agent indicated for the relief of pain in patients who require opioid analgesics for more than a few days. Morphine interacts predominantly with the opioid mu-receptor. These mu-binding sites are discretely distributed in the human brain, with high densities in the posterior amygdala, hypothalamus, thalamus, nucleus caudatus, putamen, and certain cortical areas. They are also found on the terminal axons of primary afferents within laminae I and II (substantia gelatinosa) of the spinal cord and in the spinal nucleus of the trigeminal nerve. In clinical settings, morphine exerts its principal pharmacological effect on the central nervous system and gastrointestinal tract. Its primary actions of therapeutic value are analgesia and sedation. Morphine appears to increase the patient's tolerance for pain and to decrease discomfort, although the presence of the pain itself may still be recognized. In addition to analgesia, alterations in mood, euphoria and dysphoria, and drowsiness commonly occur. Opioids also produce respiratory depression by direct action on brain stem respiratory centers.
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| Metabolism |
Morphine¿¡ ´ëÇÑ Metabolism Á¤º¸ # Phase_1_Metabolizing_Enzyme:Cytochrome P450 2D6 (CYP2D6)Catechol O-methyltransferase (COMT)
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| Absorption |
Morphine¿¡ ´ëÇÑ Absorption Á¤º¸ Bioavailability is approximately 30%.
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| Toxicity |
Morphine¿¡ ´ëÇÑ Toxicity Á¤º¸ LD50 = 461 mg/kg (rat, oral), 600 mg/kg (mouse, oral). Human lethal dose by ingestion is 120-250 mg of morphine sulfate. Symptoms of overdose include cold, clammy skin, flaccid muscles, fluid in the lungs, lowered blood pressure, "pinpoint" or dilated pupils, sleepiness leading to stupor and coma, slowed breathing, and slow pulse rate.
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| Drug Interactions |
Morphine¿¡ ´ëÇÑ Drug_Interactions Á¤º¸ Cimetidine Cimetidine increases the effect of the narcoticNaltrexone Naltrexone may precipitate a withdrawal syndrome in opioid-dependent individualsRifampin Rifampin decreases the effect of morphine/codeineTrovafloxacin IV morphine decreases the absorption of trovafloxacin
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CYP450 Drug Interaction |
[CYP450 TableÁ÷Á¢Á¶È¸]
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| Food Interaction |
Morphine¿¡ ´ëÇÑ Food Interaction Á¤º¸ Avoid alcohol.Take with food.To avoid constipation: increase your daily intake of fiber (beans, whole grains, vegetables).
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| Drug Target |
[Drug Target]
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| Description |
Morphine¿¡ ´ëÇÑ Description Á¤º¸ The principal alkaloid in opium and the prototype opiate analgesic and narcotic. Morphine has widespread effects in the central nervous system and on smooth muscle. [PubChem]
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| Drug Category |
Morphine¿¡ ´ëÇÑ Drug_Category Á¤º¸ AnalgesicsAnalgesics, OpioidNarcoticsOpiate Agonists
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| Smiles String Canonical |
Morphine¿¡ ´ëÇÑ Smiles_String_canonical Á¤º¸ CN1CCC23C4OC5=C(O)C=CC(CC1C2C=CC4O)=C35
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| Smiles String Isomeric |
Morphine¿¡ ´ëÇÑ Smiles_String_isomeric Á¤º¸ CN1CC[C@]23[C@H]4OC5=C(O)C=CC(C[C@@H]1[C@@H]2C=C[C@@H]4O)=C35
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| InChI Identifier |
Morphine¿¡ ´ëÇÑ InChI_Identifier Á¤º¸ InChI=1/C17H19NO3/c1-18-7-6-17-10-3-5-13(20)16(17)21-15-12(19)4-2-9(14(15)17)8-11(10)18/h2-5,10-11,13,16,19-20H,6-8H2,1H3/t10-,11+,13-,16-,17-/m0/s1
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| Chemical IUPAC Name |
Morphine¿¡ ´ëÇÑ Chemical_IUPAC_Name Á¤º¸ (5¥á,6¥á)-Didehydro-4,5-epoxy-17-methylmorphinan-3,6-diol
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| Drug-Induced Toxicity Related Proteins |
MORPHINE ÀÇ Drug-Induced Toxicity Related ProteinÁ¤º¸ Replated Protein:Mu-type opioid receptor Drug:Morphine Toxicity:epinephrine-induced cardiac arrhythmias. [¹Ù·Î°¡±â]
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ÀüÈ: 02-3486-1061 ¤Ó À̸ÞÀÏ: webmaster@druginfo.co.kr
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